NaV1.5 Late Current
Cell lines available: CHO and HEK293, constitutive expression. Assays validated for manual and automated patch-clamp.
Reference
|
IC50 value Peak (µM)
|
IC50 value Late (µM)
|
Flecainide
|
43.08
|
0.23
|
Lidocaine
|
446.01
|
16.88
|
Mexiletine
|
48.49
|
11.94
|
Ranolazine
|
93.85
|
18.51
|
TTX
|
2.34
|
1.09
|