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NaV1.5
Cell lines available: CHO, constitutive expression. Assays validated for manual and automated patch-clamp.
Manual patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
Propafenone |
1.6 |
Carbamazepine |
59.2 |
Quinidine |
13.6 |
TTX |
6.0 |
Automated patch-clamp (state dependent screening):
|
IC50 value (µM) |
|
IC50 value (µM) |
Resting 3rd |
5.5 |
Fast inactivated |
3.7 |
Slow inactivated |
2.7 |
|
|