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KV1.5 (IKur)
Cell lines available: CHO, constitutive expression. Assays validated for manual and automated patch-clamp.
Manual patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
Nifedipine |
45.5 |
Terfenadine |
2.9 |
Automated patch-clamp:
|
IC50 value (µM) |
Verapamil |
6.1 |