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Kir2.1
Cell lines available: CHO, constitutive expression. Assays validated for manual and automated patch-clamp.
Manual patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
ML 133 HCl pH 7.4 |
2.7 |
ML 133 HCl pH 8.5 |
0.3 |
Automated patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
ML 133 HCl pH 7.4 |
3.8 |
ML 133 HCl pH 8.5 |
0.3 |