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hERG (IKr)
Cell lines available: HEK293 / CHO, constitutive / inducible expression. Assays validated for manual and automated patch-clamp.
GLP validated assay.
Manual patch-clamp:
|
IC50 value |
|
IC50 value |
E-4031 |
11.6 nM |
Terfenadine |
15.8 nM |
Dofetelide |
11.7 nM |
Ketokonazole |
5.5 µM |
Flecainide | 1.9 nM | Cisapride | 7.3 nM |
Amiodarone | 0.2 µM | Haloperidol | 19.5 nM |
Automated patch-clamp:
|
IC50 value (µM) |
Verapamil |
0.8 |